Misoprostol
Product Name: MisoprostolSubtitle: Biological Activity: Biological Activity of MisoprostolCytoprotective prostaglandin E1 analog that displays agonist activity at EP receptors. Ki values are 120, 250, 67 and 67 nM at cloned…
Ciclesonide
Product Name: CiclesonideSubtitle: Biological Activity: SMLES: N/ACAS NO: 943764-99-6Standard In CHIKey: LUKZNWIVRBCLON-GXOBDPJESA-NMNK inhibitorsStandard InChI: InChI=1S/C32H44O7/c1-18(2)28(36)37-17-25(35)32-26(38-29(39-32)19-8-6-5-7-9-19)15-23-22-11-10-20-14-21(33)12-13-30(20,3)27(22)24(34)16-31(23,32)4/h12-14,18-19,22-24,26-27,29,34H,5-11,15-17H2,1-4H3/t22-,23-,24-,26+,27+,29+,30-,31-,32+/m0/s1Typrof Compound: Appearance: Formula: C32H44O7M.Wt: 540.69General Tips: For obtaining a higher solubility , please warm the…
UK 14,304
Product Name: UK 14,304Subtitle: Biological Activity: Biological Activity of UK 14,304Full α2 adrenergic agonist. Centrally active following systemic administration in vivo. Also available as part of the α2-Adrenoceptor and Mixed…
Dihydroergotamine mesylate
Product Name: Dihydroergotamine mesylateSubtitle: Biological Activity: Biological Activity of Dihydroergotamine mesylatePartial α-adrenergic agonist. Partial D2 dopaminergic receptor agonist. Competitive 5-HT antagonist.SMLES: N/ACAS NO: 7083-71-8Standard In CHIKey: ADYPXRFPBQGGAH-UMYZUSPBSA-NMEK inhibitorsStandard InChI: InChI=1S/C33H37N5O5.CH4O3S/c1-32(35-29(39)21-15-23-22-10-6-11-24-28(22)20(17-34-24)16-25(23)36(2)18-21)31(41)38-26(14-19-8-4-3-5-9-19)30(40)37-13-7-12-27(37)33(38,42)43-32;1-5(2,3)4/h3-6,8-11,17,21,23,25-27,34,42H,7,12-16,18H2,1-2H3,(H,35,39);1H3,(H,2,3,4Typrof…
Nicergoline
Product Name: NicergolineSubtitle: Biological Activity: Biological Activity of Nicergolineα-adrenergic, vasodilator. Cognitive enhancer.SMLES: N/ACAS NO: 23599-69-1Standard In CHIKey: YSEXMKHXIOCEJA-FVFQAYNVSA-OMAPKAPK2 MK2) inhibitorsStandard InChI: InChI=1S/C24H26BrN3O3/c1-27-13-17-8-21-24(30-3,19-5-4-6-20(27)22(17)19)9-15(12-28(21)2)14-31-23(29)16-7-18(25)11-26-10-16/h4-7,10-11,13,15,21H,8-9,12,14H2,1-3H3/p+1/t15-,21-,24+/m1/s1Typrof Compound: Appearance: Formula: C24H26BrN3O3M.Wt: 484.39General Tips: For obtaining…
SB-334867 free base
Product Name: SB-334867 free baseSubtitle: orexin-1 receptor antagonist, selectiveBiological Activity: Biological Activity of SB-334867 free baseSelective non-peptide orexin OX1 receptor antagonist. pKb values are 7.2 and < 5 for inhibition…
AMD 3465 hexahydrobromide
Product Name: AMD 3465 hexahydrobromideSubtitle: Biological Activity: Biological Activity of AMD 3465 hexahydrobromidePotent, selective CXCR4 antagonist; exhibits 8-fold higher affinity than AMD 3100. Inhibits SDF-1α-ligand binding (Ki = 41.7 nM).…
AMD 3465
Product Name: AMD 3465Subtitle: CXCR4 antagonist,potent and selectiveBiological Activity: SMLES: CAS NO: 1138245-13-2Standard In CHIKey: ERK inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C24H38N6M.Wt: 410.6General Tips: For obtaining a higher solubility…
Guanfacine
Product Name: GuanfacineSubtitle: Biological Activity: SMLES: C1=CC(=C(C(=C1)Cl)CC(=O)N=C(N)N)ClCAS NO: 1448232-80-1Standard In CHIKey: DGFYECXYGUIODH-UHFFFAOYSA-NMAPK_ERK Pathway inhibitorsStandard InChI: InChI=1S/C9H9Cl2N3O.ClH/c10-6-2-1-3-7(11)5(6)4-8(15)14-9(12)13;/h1-3H,4H2,(H4,12,13,14,15);1HTyprof Compound: Appearance: Formula: C9H9Cl2N3OM.Wt: 246.09General Tips: For obtaining a higher solubility , please warm…
Almorexant hydrochloride
Product Name: Almorexant hydrochlorideSubtitle: OX1R/OX2R antagonistBiological Activity: Biological Activity of Almorexant hydrochlorideDescription Almorexant HCl is an orally active, dual antagonist of orexin receptor with IC50 of 6.6 nM and 3.4…