Product Name: AdipoRonSubtitle: AdipoR1 and AdipoR2 agonist, first orally activeBiological Activity: SMLES: CAS NO: 194798-83-9Standard In CHIKey: Oxytocin Receptor inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C27H28N2O3M.Wt: 428.52General Tips: For obtaining…
Product Name: Montelukast SodiumSubtitle: Leukotriene receptor antagonistBiological Activity: Biological Activity of Montelukast SodiumCysteinyl leukotriene receptor 1 (CysLT1) and GPR17 antagonist. Blocks pentylenetetrazole-induced seizures, blood brain barrier (BBB) disruption and leukocyte…
Product Name: MethyldopaSubtitle: Biological Activity: Biological Activity of MethyldopaL-aromatic amino acid decarboxylase inhibitor. Antihypertensive.SMLES: CC(CC1=CC(=C(C=C1)O)O)(C(=O)O)NCAS NO: 1448169-71-8Standard In CHIKey: CJCSPKMFHVPWAR-JTQLQIEISA-NOpioid Receptor inhibitorsStandard InChI: InChI=1S/C10H13NO4/c1-10(11,9(14)15)5-6-2-3-7(12)8(13)4-6/h2-4,12-13H,5,11H2,1H3,(H,14,15)/t10-/m0/s1Typrof Compound: Appearance: Formula: C10H13NO4M.Wt: 211.21General Tips:…
Product Name: Eprosartan MesylateSubtitle: Biological Activity: SMLES: CCCCC1=NC=C(N1CC2=CC=C(C=C2)C(=O)O)C=C(CC3=CC=CS3)C(=O)O.CS(=O)(=O)OCAS NO: 887603-94-3Standard In CHIKey: DJSLTDBPKHORNY-XMMWENQYSA-NNeurotensin Receptor inhibitorsStandard InChI: InChI=1S/C23H24N2O4S.CH4O3S/c1-2-3-6-21-24-14-19(12-18(23(28)29)13-20-5-4-11-30-20)25(21)15-16-7-9-17(10-8-16)22(26)27;1-5(2,3)4/h4-5,7-12,14H,2-3,6,13,15H2,1H3,(H,26,27)(H,28,29);1H3,(H,2,3,4)/b18-12+;Typrof Compound: Appearance: Formula: C24H28N2O7S2M.Wt: 520.62General Tips: For obtaining a higher solubility , please…
Product Name: BosentanSubtitle: Biological Activity: SMLES: CC(C)(C)C1=CC=C(C=C1)S(=O)(=O)NC2=C(C(=NC(=N2)C3=NC=CC=N3)OCCO)OC4=CC=CC=C4OCCAS NO: 848258-31-1Standard In CHIKey: GJPICJJJRGTNOD-UHFFFAOYSA-NNeuropeptide Y Receptor inhibitorsStandard InChI: InChI=1S/C27H29N5O6S/c1-27(2,3)18-10-12-19(13-11-18)39(34,35)32-23-22(38-21-9-6-5-8-20(21)36-4)26(37-17-16-33)31-25(30-23)24-28-14-7-15-29-24/h5-15,33H,16-17H2,1-4H3,(H,30,31,32)Typrof Compound: Appearance: Formula: C27H29N5O6SM.Wt: 551.63General Tips: For obtaining a higher solubility , please…
Product Name: CTEP (RO4956371)Subtitle: MGlu5 inhibitorBiological Activity: Biological Activity of CTEP (RO4956371)Description CTEP (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM.…
Product Name: VU 0357121Subtitle: Biological Activity: Biological Activity of VU 0357121Positive allosteric modulator of mGlu5 receptors (EC50 = 33 nM). Binds to a site distinct from that bound by MPEP.SMLES:…
Product Name: MPEPSubtitle: MGlu5 receptor antagonistBiological Activity: SMLES: CC1=CC=CC(=N1)C#CC2=CC=CC=C2CAS NO: 16858-02-9Standard In CHIKey: Melatonin Receptor inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C14H11NM.Wt: 193.24General Tips: For obtaining a higher solubility ,…
Product Name: Ki16198Subtitle: LPA antagonistBiological Activity: SMLES: CC1=NOC(=C1NC(=O)OC(C)C2=CC=CC=C2Cl)C3=CC=C(C=C3)CSCCC(=O)OCCAS NO: 85375-15-1Standard In CHIKey: mAChR inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C24H25ClN2O5SM.Wt: 488.98General Tips: For obtaining a higher solubility , please warm…
Product Name: OC000459Subtitle: Antagonist of D prostanoid receptor 2 ,potent and selectiveBiological Activity: Biological Activity of OC000459Description OC000459 is a potent and selective antagonist of D prostanoid receptor 2 (DP2)…