Product Name: G-15
Subtitle: GPR30 antagonist, selective
Biological Activity: Biological Activity of G-15High affinity and selective GPER receptor antagonist (Ki = 20 nM) that displays no affinity for ERα and ERβ at concentrations up to 10 μM. Inhibits agonist-induced calcium mobilization in vitro (EC50 of ~185 nM) a
SMLES: BrC1=C(C=C2OCOC2=C1)[C@@H]3NC4=CC=CC=C4[C@@H]5[C@H]3CC=C5
CAS NO: 128446-36-6
Standard In CHIKey: 5 alpha Reductase inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C19H16BrNO2
M.Wt: 370.24
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/261/1/154
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 50 mM in DMSO
Storage: Store at -20℃
Purity: >98%
Chemical Name: (3aS*,4R*,9bR*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-3H-cyclopenta[c]quinoline