Product Name: GSK1324726A
Subtitle: BET proteins inhibitor
Biological Activity: Biological Activity of GSK1324726ADescription GSK1324726A is a selective small-molecule inhibitor of BET proteins with IC50 values of 41 nM, 31 nM and 22 nM for BRD2, BRD3 and BRD4, respectively . Targets BRD2 BRD3 BRD4 IC50 41 nM 3
SMLES: OC(C(C=C1)=CC=C1C2=CC3=C(C=C2)N(C(C)=O)[C@@H](C)C[C@H]3NC4=CC=C(Cl)C=C4)=O
CAS NO: 298708-79-9
Standard In CHIKey: Trk Receptor inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C25H23ClN2O3
M.Wt: 434.91
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/261/3/1064
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO
Storage:
Purity: >98%
Chemical Name: 5-[4-[[6-(4-methylsulfonylphenyl)pyridin-3-yl]oxymethyl]piperidin-1-yl]-3-propan-2-yl-1,2,4-oxadiazole