Product Name: TC-E 5003
Subtitle: PRMT1 inhibitor, potent
Biological Activity: Biological Activity of TC-E 5003Selective protein arginine methyltransferase 1 (PRMT1) inhibitor (IC50 = 1.5 μM); exhibits no inhibitory activity against CARM1 and Set7/9 methyltransferases. Inhibits growth of MCF7a breast cancer cells and LNCaP pros
SMLES: ClCC(NC1=CC=C(C=C1)S(=O)(C(C=C2)=CC=C2NC(CCl)=O)=O)=O
CAS NO: 196808-85-2
Standard In CHIKey: SHRCVZJKZJGIHQ-UHFFFAOYSA-NInfluenza Virus inhibitors
Standard InChI: InChI=1S/C16H14Cl2N2O4S/c17-9-15(21)19-11-1-5-13(6-2-11)25(23,24)14-7-3-12(4-8-14)20-16(22)10-18/h1-8H,9-10H2,(H,19,21)(H,20,22)
Typrof Compound:
Appearance:
Formula: C16H14Cl2N2O4S
M.Wt: 401.26
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/262/1/271
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 50 mM in DMSO
Storage: Store at +4℃
Purity: >98%
Chemical Name: N,N'-(Sulfonyldi-4,1-phenylene)bis(2-chloroacetamide)