Product Name: 3-pyr-Cytisine
Subtitle: α4β2 receptors agonist
Biological Activity: Biological Activity of 3-pyr-CytisineHigh affinity α4β2 partial agonist (Ki values are 0.91, 119 and 1100 nM for α4β2, α3β4 and α7 receptors respectively). Shows little activity at α3β4 and α7 receptors. E
SMLES:
CAS NO: 4044-65-9
Standard In CHIKey: CNS-penetrant_Compound_Library inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C16H17N3O
M.Wt: 267.33
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/269/2/659
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in water and to 100 mM in DMSO
Storage: Store at -20℃
Purity: >98%
Chemical Name: (1R,5S)-1,2,3,4,5,6-Hexahydro-9-(3-pyridinyl)-1,5-methano-8H-pyrido[1,2-a][1,5]diazocin-8-one