Product Name: A 438079 hydrochloride
Subtitle: P2X7 receptor antagonist,competitive and selective
Biological Activity: Biological Activity of A 438079 hydrochlorideCompetitive P2X7 receptor antagonist (pIC50 = 6.9 for the inhibition of Ca2+ influx in the human recombinant P2X7 cell line). Devoid of activity at other P2 receptors (IC50 >> 10 μM). Possesses antinoc
SMLES:
CAS NO: 1032350-13-2
Standard In CHIKey: Polo-like Kinase PLK) inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C13H10Cl3N5
M.Wt: 342.61
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/258/2/626
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 5 mM in water with gentle warming and to 100 mM in DMSO
Storage: Desiccate at RT
Purity: >98%
Chemical Name: 3-[[5-(2,3-Dichlorophenyl)-1H-tetrazol-1-yl]methyl]pyridine hydrochloride