Product Name: A 80426 mesylate
Subtitle: α2-adrenoceptor antagonist and 5-HT uptake inhibitor
Biological Activity: Biological Activity of A 80426 mesylateHigh affinity α2-adrenoceptor antagonist and selective 5-HT uptake inhibitor (Ki values are 2.01 and 3.77 nM respectively). Displays low affinity at a variety of structurally homologous GPCRs.
SMLES:
CAS NO: 92169-45-4
Standard In CHIKey: NF-kappa)B inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C23H27NO2.CH3SO3H
M.Wt: 445.57
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/265/2/813
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 10 mM in water and to 100 mM in DMSO
Storage: Desiccate at +4℃
Purity: >98%
Chemical Name: N-Methyl-N-[[(1R)-1,2,3,4-tetrahydro-5-methoxy-1-naphthalenyl]methyl]-6-benzofuranethanamine mesylate