Product Name: A-867744
Subtitle: Allosteric Modulator
Biological Activity: Biological Activity of A-867744Positive allosteric modulator of α7 nAChRs (IC50 values are 0.98 and 1.12 μM for human and rat α7 receptor ACh-evoked currents respectively, in X. laevis oocytes). Displays no activity at 5-HT3A, α3β
SMLES:
CAS NO: 174022-42-5
Standard In CHIKey: Anti-virus_Compound_Library inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C20H19ClN2O3S
M.Wt: 402.89
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/256/3/954
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO and to 10 mM in ethanol with gentle warming
Storage: Store at +4℃
Purity: >98%
Chemical Name: 4-[5-(4-Chlorophenyl)-2-methyl-3-(1-oxopropyl)-1H-pyrrol-1-yl]benzenesulfonamide