Product Name: BMS 470539 dihydrochloride
Subtitle: MC1 receptor,potent and selective
Biological Activity: Biological Activity of BMS 470539 dihydrochloridePotent, selective melanocortin MC1 receptor agonist (IC50 = 120 nM). Exhibits anti-inflammatory properties following ischemia-reperfusion in the vasculature. Inhibits leukocyte trafficking.
SMLES:
CAS NO: 80321-63-7
Standard In CHIKey: Cell Cycle_DNA Damage inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C32H41N5O4.2HCl
M.Wt: 632.62
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/266/1/74
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in water and to 100 mM in DMSO
Storage: Desiccate at RT
Purity: >98%
Chemical Name: 1-[1-(3-Methyl-L-histidyl-O-methyl-D-tyrosyl)-4-phenyl-4-piperidinyl]-1-butanone dihydrochloride