Product Name: BMS-509744
Subtitle: Itk inhibitor,potent and selective
Biological Activity: Biological Activity of BMS-509744Potent and selective interleukin-2 inducible T cell kinase (ITK) inhibitor (IC50 = 19 nM). Displays 200-fold selectivity over Tec family kinases and 55-fold selectivity over other kinases tested. Reduces HIV infection of p
SMLES:
CAS NO: 208255-80-5
Standard In CHIKey: nAChR inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C32H41N5O4S2
M.Wt: 623.83
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/259/1/430
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in 1eq. HCl and to 50 mM in DMSO
Storage: Store at -20℃
Purity: >98%
Chemical Name: N-[5-[[5-[(4-Acetyl-1-piperazinyl)carbonyl]-4-methoxy-2-methylphenyl]thio]-2-thiazolyl]-4-[[(1,2,2-trimethylpropyl)amino]methyl]benzamide