Product Name: BRL-15572
Subtitle: 5-HT1D receptor antagonist
Biological Activity: Biological Activity of BRL-15572Description BRL-15572 is an antagonist of 5-HT1D receptor with a pKi value of 7.9. Targets 5-HT1D 5-HT1A 5-HT2B 5-HT2A 5-HT7 IC50 7.9(pKi) 7.7(pKi) 7.4(pKi) 6.6(pKi) 6.3(pKi)
SMLES: C1CN(CCN1CC(C(C2=CC=CC=C2)C3=CC=CC=C3)O)C4=CC(=CC=C4)Cl.Cl.Cl
CAS NO: 3485-62-9
Standard In CHIKey: Keap1-Nrf2 inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C25H27ClN2O.ClH.ClH
M.Wt: 478.13
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/269/1/193
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: 3-[4-(3-chlorophenyl)piperazin-1-yl]-1,1-diphenylpropan-2-ol;dihydrochloride