Product Name: CAL-101 (Idelalisib, GS-1101)
Subtitle: PI3K inhibitor
Biological Activity: Biological Activity of CAL-101 (Idelalisib, GS-1101)Description CAL-101 (Idelalisib, GS-1101) is a selective inhibitor of p110δ with IC50 of 2.5 nM. Targets p110δ IC50 2.5 nM
SMLES: CCC(C1=NC2=C(C(=CC=C2)F)C(=O)N1C3=CC=CC=C3)NC4=NC=NC5=C4NC=N5
CAS NO: 147127-20-6
Standard In CHIKey: ADC Linker inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C22H18FN7O
M.Wt: 415.43
General Tips: for obtaining a higher concentration: Please warm the tube at 37 °C for 10 minutes and/or shake it in the ultrasonic bath for a while.Stock solution can be stored below -20°C for several months.PubMed ID:http://jpet.aspetjournals.org/content/257/1/457
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: 5-fluoro-3-phenyl-2-[(1S)-1-(7H-purin-6-ylamino)propyl]quinazolin-4-one