Product Name: EHT 1864
Subtitle: Rac family small GTPases inhibitor
Biological Activity: Biological Activity of EHT 1864Inhibitor of Rac family GTPases. Blocks activation by direct binding to Rac1, Rac1b, Rac2 and Rac3 (KD values are 40, 50, 60 and 250 nM respectively). Inhibits Rac, Ras and Tiam-induced growth transformation of NIH-3T3 fibr
SMLES: CCN1C2=C(C=C(C=C2)NC3=NC(=NC=C3)NCCCN4CCOCC4)C5=CC=CC=C51
CAS NO: 302-22-7
Standard In CHIKey: Apoptosis_Compound_Library inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C25H29Cl2F3N2O4S
M.Wt: 581.48
General Tips: for obtaining a higher concentration: Please warm the tube at 37 ℃ for 10 minutes and/or shake it in the ultrasonic bath for a while. Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/269/2/632
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in water and to 75 mM in DMSO
Storage: Store at +4℃
Purity: >98%
Chemical Name: 5-(5-(7-(Trifluoromethyl)quinolin-4-ylthio)pentyloxy)-2-(morpholinomethyl)-4H-pyran-4-one dihydrochloride