Product Name: GR 127935 hydrochloride
Subtitle:
Biological Activity: Biological Activity of GR 127935 hydrochloridePotent and selective 5-HT1B/1D receptor antagonist (pKi values are 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptors). Displays > 100-fold selectivity over 5HT1A, 5-HT2A, 5-HT2C receptors and other re
SMLES: O=C(C(C=C1)=CC=C1C2=CC=C(C3=NOC(C)=N3)C=C2C)NC4=CC=C(C(N5CCN(C)CC5)=C4)OC.Cl
CAS NO: 1334298-90-6
Standard In CHIKey: Potassium Channel inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C29H31N5O3.HCl
M.Wt: 534.06
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/265/1/321
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in water
Storage: Desiccate at RT
Purity: >98%
Chemical Name: N-[4-Methoxy-3-(4-methyl-1-piperazinyl)phenyl]-2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)-1,1-biphenyl-4-carboxamide hydrochloride

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