Product Name: GS 39783
Subtitle:
Biological Activity: Biological Activity of GS 39783Positive allosteric modulator of GABAB receptor function. Potentiates the effects of GABA on [35S]GTPγS binding at recombinant and native GABAB receptors (EC50 values are 2.1 and 3.1μM respectively). Decreases cocai
SMLES: [O-][N+](C1=C(N=C(N=C1NC2CCCC2)SC)NC3CCCC3)=O
CAS NO: 1134156-31-2
Standard In CHIKey: IGF-1R inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C15H23N5O2S
M.Wt: 337.44
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/273/3/1471
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 5 mM in ethanol and to 10 mM in DMSO
Storage: Store at RT
Purity: >98%
Chemical Name: N,N-Dicyclopentyl-2-(methylthio)-5-nitro-4,6-pyrimidinediamine