Product Name: GSK343
Subtitle: EZH2 inhibitor,potent,selective and cell permeable
Biological Activity: Biological Activity of GSK343Description GSK343 is a cell-permeable inhibitor of EZH2 with IC50 value of 4 nM. Targets EZH2 IC50 4 nM
SMLES: CCCC1=C(C(=O)NC(=C1)C)CNC(=O)C2=C3C=NN(C3=CC(=C2)C4=CC(=NC=C4)N5CCN(CC5)C)C(C)C
CAS NO: 1032229-33-6
Standard In CHIKey: Procollagen C Proteinase inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C31H39N7O2
M.Wt: 541.69
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/259/2/799
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Limited solubility
Storage:
Purity: >98%
Chemical Name: N-[(6-methyl-2-oxo-4-propyl-1H-pyridin-3-yl)methyl]-6-[2-(4-methylpiperazin-1-yl)pyridin-4-yl]-1-propan-2-ylindazole-4-carboxamide