Product Name: GW 803430
Subtitle:
Biological Activity: Biological Activity of GW 803430Selective melanin-concentrating hormone receptor 1 (MCH1) antagonist (IC50 = 9.3 nM). Displays antiobesity and antidepressant-like effects in rats and mice. Orally active.
SMLES: ClC1=CC=C(C=C1)C2=CC(N=CN(C3=O)C4=CC=C(C(OC)=C4)OCCN5CCCC5)=C3S2
CAS NO: 1370468-36-2
Standard In CHIKey: DNA-PK inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C25H24ClN3O3S
M.Wt: 481.99
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/266/2/1066
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 25 mM in 1eq. HCl
Storage: Store at +4℃
Purity: >98%
Chemical Name: 6-(4-Chlorophenyl)-3-[3-methoxy-4-[2-(1-pyrrolidinyl)ethoxy]phenyl]-thieno[3,2-d]pyrimidin-4(3H)-one