Product Name: H 89 2HCl
Subtitle: Potent PKA inhibitor
Biological Activity: Biological Activity of H 89 2HClProtein kinase A inhibitor that also inhibits several other kinases (IC50 values are 80, 120, 135, 270, 2600 and 2800 nM for S6K1, MSK1, PKA, ROCKII, PKBα and MAPKAP-K1b). Exhibits antinociceptive activity. Also avail
SMLES: O=S(C1=CC=CC2=C1C=CN=C2)(NCCNC/C=C/C3=CC=C(Br)C=C3)=O.Cl.Cl
CAS NO: 338967-87-6
Standard In CHIKey: Kinesin inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C20H20BrN3O2S.2HCl
M.Wt: 519.28
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/255/2/549
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 25 mM in water and to 100 mM in DMSO
Storage: Store at -20℃
Purity: >98%
Chemical Name: N-[2-[[3-(4-Bromophenyl)-2-propenyl]amino]ethyl]-5-isoquinolinesulfonamide dihydrochloride