Product Name: L-838,417
Subtitle:
Biological Activity: Biological Activity of L-838,417Subtype-selective GABAA receptor partial agonist. Selectively binds to α1, α2, α3 and α5 subunits (Ki values are 0.79, 0.67, 0.67 and 2.25 nM respectively) but displays no efficacy at α1 (α1-sp
SMLES: FC(C(C1=NN=C2N1N=C(C(C(C)(C)C)=C2)OCC3=NC=NN3C)=C4)=CC=C4F
CAS NO: 1146963-51-0
Standard In CHIKey: Others inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C19H19F2N7O
M.Wt: 399.4
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/274/1/584
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO and to 20 mM in ethanol with sonication
Storage: Store at +4℃
Purity: >98%
Chemical Name: 3-(2,5-Difluorophenyl)-7-(1,1-dimethylethyl)-6-[(1-methyl-1H-1,2,4-triazol-5-yl)methoxy]-1,2,4-triazolo[4,3-b]pyridazine