Product Name: LY 215840
Subtitle:
Biological Activity: Biological Activity of LY 2158405-HT2/5-HT7 receptor antagonist. Reduces stimulatory effect of serotonin on aldosterone secretion; also reduces 5-HT-induced cAMP formation (pKB = 8.26).
SMLES: O=C([C@@H]1C[C@@H]2[C@@H](CC3=CN(C(C)C)C4=CC=CC2=C34)N(C)C1)N[C@@H](CCC5)[C@@H]5O
CAS NO: 69-33-0
Standard In CHIKey: IMSDOBUYDTVEHN-LUKLFJNJSA-NMetabolic Enzyme_Protease inhibitors
Standard InChI: InChI=1S/C24H33N3O2/c1-14(2)27-13-15-11-21-18(17-6-4-8-20(27)23(15)17)10-16(12-26(21)3)24(29)25-19-7-5-9-22(19)28/h4,6,8,13-14,16,18-19,21-22,28H,5,7,9-12H2,1-3H3,(H,25,29)/t16-,18?,19+,21-,22-/m1/s1
Typrof Compound:
Appearance:
Formula: C24H33N3O2
M.Wt: 395.54
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/265/1/366
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO and to 25 mM in ethanol
Storage: Store at +4℃
Purity: >98%
Chemical Name: [8β(1S,2R)]-N-(2-Hydroxycyclopentyl)-6-methyl-1-(1-methylethyl)-ergoline-8-carboxamide