Product Name: MLN2238
Subtitle: β5 site of the 20S proteasome inhibitor
Biological Activity: Biological Activity of MLN2238Description MLN2238 is an inhibitor of the chymotrypsin-like proteolytic (β5) site of the 20S proteasome with IC50 and Ki values of 3.4 nM and 0.93 nM, also inhibitor of the caspase-like (β1) and trypsin-like (β2) proteolyt
SMLES: B(C(CC(C)C)NC(=O)CNC(=O)C1=C(C=CC(=C1)Cl)Cl)(O)O
CAS NO: 343787-29-1
Standard In CHIKey: Androgen Receptor inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C14H19BCl2N2O4
M.Wt: 361
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/259/3/997
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: [(1R)-1-[[(2S,3R)-3-hydroxy-2-[(6-phenylpyridine-2-carbonyl)amino]butanoyl]amino]-3-methylbutyl]boronic acid

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