Product Name: MRS 1754
Subtitle:
Biological Activity: Biological Activity of MRS 1754Selective adenosine A2B receptor antagonist (Ki values are 1.97, 16.8, 403, 503, 570 and 612 nM for hA2B, rA1, hA1, hA2A, hA3 and rA2A receptors respectively).
SMLES: O=C(N(C1=O)CCC)N(CCC)C2=C1NC(C(C=C3)=CC=C3OCC(NC4=CC=C(C#N)C=C4)=O)=N2
CAS NO: 871361-88-5
Standard In CHIKey: beta)-catenin inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C26H26N6O4
M.Wt: 486.52
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/265/3/1232
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 5 mM in DMSO with gentle warming and to 10 mM in DMSO with sonication
Storage: Desiccate at RT
Purity: >98%
Chemical Name: N-(4-Cyanophenyl)-2-[4-(2,3,6,7-tetrahydro-2,6-dioxo-1,3-dipropyl-1H-purin-8-yl)phenoxy]-acetamide