Product Name: Nepicastat
Subtitle: Inhibitor of dopamine-β-hydroxylase,potent and selective
Biological Activity: Biological Activity of NepicastatDescription Nepicastat is a selective inhibitor of dopamine β-hydroxylase (DBH) with IC50 value of 9 nM. Targets DBH IC50 9 nM
SMLES: C1CC2=C(C=C(C=C2CC1N3C(=CNC3=S)CN)F)F
CAS NO: 459789-99-2
Standard In CHIKey: YZZVIKDAOTXDEB-UHFFFAOYSA-OROR inhibitors
Standard InChI: InChI=1S/C14H15F2N3S/c15-9-3-8-4-10(1-2-12(8)13(16)5-9)19-11(6-17)7-18-14(19)20/h3,5,7,10H,1-2,4,6,17H2,(H,18,20)/p+1
Typrof Compound:
Appearance:
Formula: C14H15F2N3S
M.Wt: 295.35
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/254/2/393
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: DMSO
Storage:
Purity: >98%
Chemical Name: 4-(aminomethyl)-3-[(2S)-5,7-difluoro-1,2,3,4-tetrahydronaphthalen-2-yl]-1H-imidazole-2-thione