Product Name: ONO-AE3-208
Subtitle: EP4 receptor inhibitor,high affinity and selective
Biological Activity: Biological Activity of ONO-AE3-208High affinity and selective EP4 receptor antagonist (Ki values are 1.3, 30, 790 and 2400 nM for EP4, EP3, FP and TP receptors respectively). Displays no affinity for EP1, EP2, DP or IP receptors (Ki >10 μM). Inh
SMLES: O=C(Nc1cc(C#N)ccc1CCCC(=O)O)C(c3c2ccccc2c(F)cc3)C
CAS NO: 906805-42-3
Standard In CHIKey: Stearoyl-CoA Desaturase SCD) inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C24H21FN2O3
M.Wt: 404.43
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/254/2/412
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO and to 10 mM in 1.1eq. NaOH with gentle warming
Storage: Store at -20℃
Purity: >98%
Chemical Name: 4-Cyano-2-[[2-(4-fluoro-1-naphthalenyl)-1-oxopropyl]amino]benzenebutanoic acid