Product Name: Orteronel
Subtitle: For castration-resistant prostate cancer, clinical candidate
Biological Activity: Biological Activity of OrteronelDescription TAK-700 (Orteronel) is a potent and highly selective inhibitor of human and rat 17,20-lyase with IC50 values of 38 nM and 54 nM, respectively. Targets 17,20-lyase IC50 38 nM (human) 54 nM
SMLES: CNC(=O)C1=CC2=C(C=C1)C=C(C=C2)C3(CCN4C3=CN=C4)O
CAS NO: 202590-98-5
Standard In CHIKey: Thrombin inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C18H17N3O2
M.Wt: 307.35
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/254/2/420
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO
Storage:
Purity: >98%
Chemical Name: 6-[(7S)-7-hydroxy-5,6-dihydropyrrolo[1,2-c]imidazol-7-yl]-N-methylnaphthalene-2-carboxamide