Product Name: PNU 142633
Subtitle:
Biological Activity: Biological Activity of PNU 142633Very selective, high affinity 5-HT1D receptor agonist (Ki values are 6 and > 18000 nM at human 5-HT1D and 5-HT1B receptors respectively). Inhibits sympathetically-induced tachycardic responses and blocks neurogenic plas
SMLES: O=C(C1=CC2=C(C=C1)[C@H](CCN3CCN(C4=CC=C(C(N)=O)C=C4)CC3)OCC2)NC
CAS NO: 881681-00-1
Standard In CHIKey: LXR inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C24H30N4O3
M.Wt: 422.53
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/265/2/543
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO
Storage: Store at +4℃
Purity: >98%
Chemical Name: (1S)-1-[2-[4-[4-(Aminocarbonyl)phenyl]-1-piperazinyl]ethyl]-3,4-dihydro-N-methyl-1H-2-benzopyran-6-carboxamide