Product Name: PRX-08066 Maleic acid
Subtitle: 5-HT2B receptor antagonist,potent and selective
Biological Activity: Biological Activity of PRX-08066 Maleic acidDescription PRX-08066 Maleic acid is a selective antagonist of 5-HT2B receptor with IC50 value of 3.4 nM. Targets 5-HT2B IC50 3.4 nM
SMLES: c1cc(c(cc1CN2CCC(CC2)Nc3c4cc(sc4ncn3)Cl)C#N)F.C(=CC(=O)O)C(=O)O
CAS NO: 1374639-75-4
Standard In CHIKey: Cardiovascular Disease inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C19H17ClFN5S.C4H4O4
M.Wt: 517.96
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/256/3/890
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: 5-({4-[(6-Chlorothieno[2,3-d]pyrimidin-4-yl)amino]-1-piperidinyl}methyl)-2-fluorobenzonitrile (2Z)-2-butenedioate (1:1)