Product Name: Pitolisant hydrochloride
Subtitle: Nonimidazole inverse agonist
Biological Activity: Biological Activity of Pitolisant hydrochlorideHistamine H3 receptor inverse agonist (EC50 = 1.5 nM) and antagonist (Ki = 0.16 nM). Exhibits nootropic effects in cognitive disorders; reduces locomotor hyperactivity induced by methamphetamine. Brain penetr
SMLES: C1CCN(CC1)CCCOCCCC2=CC=C(C=C2)Cl.Cl
CAS NO: 9087-70-1
Standard In CHIKey: IAP inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C17H27Cl2NO
M.Wt: 332.31
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/267/3/1544
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in water and to 100 mM in DMSO
Storage: Desiccate at RT
Purity: >98%
Chemical Name: 1-[3-[3-(4-Chlorophenyl)propoxy]propyl]-piperidine hydrochloride