Product Name: Ro 15-4513
Subtitle:
Biological Activity: Biological Activity of Ro 15-4513High affinity benzodiazepine ligand. Ki values are 3.1 and 5.3 nM for diazepam-insensitive (DI) and diazepam-sensitive (DS) benzodiazepine receptors respectively. Acts as partial inverse agonist at recombinant DS α1-
SMLES: O=C1N(C)CC2=C(C(OCC)=O)N=CN2C(C1=C3)=CC=C3N=[N+]=[N-]
CAS NO: 1230487-00-9
Standard In CHIKey: CFSOJZTUTOQNIA-UHFFFAOYSA-NFAK inhibitors
Standard InChI: InChI=1S/C15H14N6O3/c1-3-24-15(23)13-12-7-20(2)14(22)10-6-9(18-19-16)4-5-11(10)21(12)8-17-13/h4-6,8H,3,7H2,1-2H3
Typrof Compound:
Appearance:
Formula: C15H14N6O3
M.Wt: 326.31
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/273/3/1442
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 5 mM in ethanol and to 10 mM in DMSO
Storage: Desiccate at +4℃
Purity: >98%
Chemical Name: 8-Azido-5,6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]benzodiazepine-3-carboxylic acid ethyl ester