Product Name: Ro 25-6981 Maleate
Subtitle: NMDA receptor antagonist,potent and selective
Biological Activity: Biological Activity of Ro 25-6981 MaleatePotent and selective activity-dependent blocker of NMDA receptors containing the NR2B subunit. IC50 values are 0.009 and 52 μM for cloned receptor subunit combinations NR1C/NR2B and NR1C/NR2A respectively. Displ
SMLES: OC1=CC=C([C@@H](O)[C@@H](C)CN2CCC(CC3=CC=CC=C3)CC2)C=C1.O=C(O)/C=CC(O)=O
CAS NO: 52705-93-8
Standard In CHIKey: DYRK inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C26H33NO6
M.Wt: 455.54
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/271/3/1462
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 10 mM in water with gentle warming and to 100 mM in DMSO
Storage: Desiccate at RT
Purity: >98%
Chemical Name: (αR,βS)-α-(4-Hydroxyphenyl)-β-methyl-4-(phenylmethyl)-1-piperidinepropanol maleate