Product Name: SB 218795
Subtitle:
Biological Activity: Biological Activity of SB 218795Potent, selective and competitive non-peptide NK3 receptor antagonist (Ki = 13 nM at hNK3). Displays 90-fold and 7000-fold selectivity over hNK2 and hNK1 receptors respectively. Active in vivo, inhibiting agonist-induced pu
SMLES: O=C(C1=CC(C2=CC=CC=C2)=NC3=CC=CC=C13)N[C@H](C(OC)=O)C4=CC=CC=C4
CAS NO: 839707-37-8
Standard In CHIKey: Monoamine Transporter inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C25H20N2O3
M.Wt: 396.44
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/265/1/263
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO and to 5 mM in ethanol
Storage: Store at RT
Purity: >98%
Chemical Name: (R)-[[2-Phenyl-4-quinolinyl)carbonyl]amino]-methyl ester benzeneacetic acid