Product Name: SB 221284
Subtitle:
Biological Activity: Biological Activity of SB 221284Potent, selective 5-HT2C/2B receptor antagonist. pKi values are 6.4, 7.9 and 8.6 for 5-HT2A, 2B and 2C receptors respectively. Centrally active upon systemic administration in vivo.
SMLES: FC(F)(C(C=C1N(C(NC2=CC=CN=C2)=O)CCC1=C3)=C3SC)F
CAS NO: 1445379-92-9
Standard In CHIKey: Monocarboxylate Transporter inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C16H14F3N3OS
M.Wt: 353.36
General Tips: For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while.Stock solution can be stored below -20℃ for several months.PubMed ID:http://jpet.aspetjournals.org/content/265/1/273
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble to 100 mM in DMSO
Storage: Store at +4℃
Purity: >98%
Chemical Name: 2,3-Dihydro-5-(methylthio)-N-3-pyridinyl-6-(trifluoromethyl)-1H-indole-1-carboxamide