Product Name: WP1130
Subtitle: Deubiquitinase (DUB) inhibitor, Cell permeable
Biological Activity: Biological Activity of WP1130Description Degrasyn (WP1130) is a selective inhibitor of deubiquitinase (DUB: USP5, UCH-L1, USP9x, USP14, and UCH37). Targets DUB Bcr-Abl IC50 1.8 μM
SMLES: CCCC(C1=CC=CC=C1)NC(=O)C(=CC2=NC(=CC=C2)Br)C#N
CAS NO: 24386-93-4
Standard In CHIKey: Infection inhibitors
Standard InChI:
Typrof Compound:
Appearance:
Formula: C19H18BrN3O
M.Wt: 384.27
General Tips: for obtaining a higher concentration: Please warm the tube at 37 °C for 10 minutes and/or shake it in the ultrasonic bath for a while.Stock solution can be stored below -20°C for several months.PubMed ID:http://jpet.aspetjournals.org/content/26/1/61
Shipping Condition: Packaging according to customer requirements(5mg, 10mg, 20mg and more). Ship via FedEx, DHL, UPS, EMS or other courier with RT , or blue ice upon request.
Solubility: Soluble in DMSO > 10 mM
Storage:
Purity: >98%
Chemical Name: (E)-3-(6-bromopyridin-2-yl)-2-cyano-N-[(1S)-1-phenylbutyl]prop-2-enamide