Product Name: SB-674042Subtitle: OX1 selective antagonistBiological Activity: Biological Activity of SB-674042Potent and selective non-peptide orexin OX1 receptor antagonist (Kd = 3.76 nM). Exhibits 100-fold selectivity for OX1 over OX2 receptors.…
Product Name: SB-408124 HydrochlorideSubtitle: OX1 receptor antagonist,selective and non-peptideBiological Activity: SMLES: N/ACAS NO: 827022-33-3Standard In CHIKey: Keap1-Nrf2 inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C19H19ClF2N4OM.Wt: 392.83General Tips: For obtaining a higher…
Product Name: SB-222200Subtitle: Human NK-3 receptor antagonistBiological Activity: Biological Activity of SB-222200Potent and selective non-peptide NK3 receptor antagonist (Ki values are 4.4, > 100,000 and 250 nM for human NK3,…
Product Name: Salmeterol xinafoateSubtitle: β2-adrenergic receptor agonistBiological Activity: Biological Activity of Salmeterol xinafoateLong-acting β2 adrenergic receptor agonist. Inhibits the release of histamine, leukotrienes and prostaglandin D2, and blocks GM-CSF production…
Product Name: SalmefamolSubtitle: Biological Activity: SMLES: CC(CC1=CC=C(C=C1)OC)NCC(C2=CC(=C(C=C2)O)CO)OCAS NO: 905579-51-3Standard In CHIKey: VPMWDFRZSIMDKW-YJYMSZOUSA-Ngamma)-secretase inhibitorsStandard InChI: InChI=1S/C19H25NO4/c1-13(9-14-3-6-17(24-2)7-4-14)20-11-19(23)15-5-8-18(22)16(10-15)12-21/h3-8,10,13,19-23H,9,11-12H2,1-2H3/t13-,19+/m1/s1Typrof Compound: Appearance: Formula: C19H25NO4M.Wt: 331.42General Tips: For obtaining a higher solubility , please warm the…
Product Name: RS 504393Subtitle: CCR2 chemokine receptor antagonistBiological Activity: Biological Activity of RS 504393Extremely selective CCR2 chemokine receptor antagonist (IC50 values are 98 nM and > 100 μM for inhibition…
Product Name: Rimonabant hydrochlorideSubtitle: CB1 receptor inverse agonistBiological Activity: Biological Activity of Rimonabant hydrochloridePotent and selective cannabinoid CB1 receptor antagonist (Ki = 1.98 nM). Also acts as an inverse agonist…
Product Name: Reparixin L-lysine saltSubtitle: CXCR1/CXCR2 inhibitorBiological Activity: SMLES: CC(C)CC1=CC=C(C=C1)C(C)C(=O)NS(=O)(=O)C.C(CCN)CC(C(=O)O)NCAS NO: 923287-50-7Standard In CHIKey: CaMK inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C20H35N3O5SM.Wt: 429.57General Tips: for obtaining a higher concentration: Please…
Product Name: ReparixinSubtitle: Inhibitor of CXCL8 receptor and CXCR1/CXCR2 activationBiological Activity: SMLES: CC(C)CC1=CC=C(C=C1)C(C)C(=O)NS(=O)(=O)CCAS NO: 273404-37-8Standard In CHIKey: KQDRVXQXKZXMHP-UHFFFAOYSA-NBeta-secretase inhibitorsStandard InChI: InChI=1S/C14H21NO3S/c1-10(2)9-12-5-7-13(8-6-12)11(3)14(16)15-19(4,17)18/h5-8,10-11H,9H2,1-4H3,(H,15,16)Typrof Compound: Appearance: Formula: C14H21NO3SM.Wt: 283.39General Tips: for obtaining a…
Product Name: PreladenantSubtitle: Adenosine A2A receptor antagonistBiological Activity: Biological Activity of PreladenantDescription Preladenant (SCH 420814) is a potent and selective antagonist of adenosine A2A receptor. Targets adenosine A2A receptor IC50SMLES:…