Product Name: NociceptinSubtitle: Biological Activity: Biological Activity of NociceptinHighly potent and selective NOP receptor agonist (EC50 = 1 nM). Displays > 875-fold selectivity over opioid receptors (IC50 values are 0.32,…
Product Name: Nociceptin(1-13)NH2Subtitle: Biological Activity: Biological Activity of Nociceptin(1-13)NH2Highly potent and selective nociceptin/orphanin FQ receptor (OP4) agonist peptide (pKi = 10.68; pEC50 = 9.80). Displays > 8000-fold selectivity over δ,…
Product Name: UFP-101Subtitle: Biological Activity: Biological Activity of UFP-101Potent, selective and competitive silent antagonist for the NOP opioid receptor. Binds to NOP with high affinity (pKi = 10.24) and displays…
Product Name: LY 288513Subtitle: Biological Activity: Biological Activity of LY 288513Selective CCK2 receptor antagonist (IC50 values are 16 and > 30,000 nM for CCK2 and CCK1 respectively). Displays anxiolytic and…
Product Name: tcY-NH2Subtitle: Biological Activity: Biological Activity of tcY-NH2Selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.SMLES: O=C((CC(C=C1)=CC=C1O)NC(/C=C/C2=CC=CC=C2)=O)N3(C(NCC(N(C(N(C(N)=O)CC4=CC=CC=C4)=O)CCCCN)=O)=O)CCC3CAS NO: 1404095-34-6Standard In CHIKey: Amyloid-beta) inhibitorsStandard InChI: Typrof…
Product Name: Proglumide sodium saltSubtitle: Biological Activity: Biological Activity of Proglumide sodium saltNon-selective cholecystokinin (CCK) antagonist. Inhibits CCK-stimulated amylase secretion and prevents CCK-induced 2-deoxyglucose uptake in mouse pancreatic acini. Blocks…
Product Name: Ghrelin (rat)Subtitle: Biological Activity: Biological Activity of Ghrelin (rat)Endogenous agonist peptide for the ghrelin receptor (GHS-R1a). Produced mainly by the stomach, it stimulates release of growth hormone from…
Product Name: Orexin B (mouse)Subtitle: Biological Activity: Biological Activity of Orexin B (mouse)Endogenous agonist at orexin receptors. May be involved in the regulation of feeding, sleep-wake cycle and other hypothalamic…
Product Name: Orexin B (human)Subtitle: Biological Activity: Biological Activity of Orexin B (human)Endogenous agonist at orexin receptors (Ki values are 420 and 36 nM for OX1 and OX2 receptors, respectively).…
Product Name: Orexin A (human, rat, mouse)Subtitle: Biological Activity: Biological Activity of Orexin A (human, rat, mouse)Endogenous agonist at orexin receptors (Ki values are 20 and 38 nM for OX1…