Product Name: CC-401Subtitle: JNK inhibitor,ATP-competitiveBiological Activity: SMLES: C1CCN(CC1)CCOC2=CC=CC(=C2)C3=NNC4=C3C=C(C=C4)C5=NC=NN5CAS NO: 229975-97-7Standard In CHIKey: DNA_RNA Synthesis inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C22H24N6OM.Wt: 388.47General Tips: For obtaining a higher solubility , please…
Product Name: LGX818Subtitle: RAF inhibitor,potent and selectiveBiological Activity: Biological Activity of LGX818Description Encorafenib (LGX818) is a highly potent inhibitor of RAF with selective anti-proliferative and apoptotic activity in cells expressing…
Product Name: B-Raf inhibitor 1 dihydrochlorideSubtitle: B-Raf inhibitor,potent and selectiveBiological Activity: Biological Activity of B-Raf inhibitor 1 dihydrochlorideDescription B-Raf inhibitor 1 dihydrochloride is a potent and selective inhibitor of B-Raf…
Product Name: B-Raf inhibitor 1Subtitle: Biological Activity: SMLES: CC1=C(C2=C(C=C1)C(=NC=C2)NC3=CC=C(C=C3)Cl)NC4=C(C=CC=N4)C5=C6C(=NC=N5)N=CN6CAS NO: 1449277-10-4Standard In CHIKey: Deubiquitinase inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C26H19ClN8M.Wt: 478.94General Tips: For obtaining a higher solubility , please…
Product Name: SB 242235Subtitle: MAPK inhibitorBiological Activity: SMLES: COC1=NC=CC(=N1)C2=C(N=CN2C3CCNCC3)C4=CC=C(C=C4)FCAS NO: 302962-49-8Standard In CHIKey: CRISPR_Cas9 inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C19H20FN5OM.Wt: 353.39General Tips: For obtaining a higher solubility , please…
Product Name: GDC-0623Subtitle: MEK1 inhibitor, potent and ATP-uncompetitiveBiological Activity: Biological Activity of GDC-0623Description GDC-0623 is a potent and ATP-uncompetitive inhibitor of MEK1 with Ki value of 0.13 nM. Targets MEK1…
Product Name: VRT752271Subtitle: ERK1/ERK2 inhibitorBiological Activity: SMLES: CC(C)NC1=NC=C(C(=C1)C2=CNC(=C2)C(=O)NC(CO)C3=CC(=CC=C3)Cl)ClCAS NO: 585543-15-3Standard In CHIKey: CDK inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C21H22Cl2N4O2M.Wt: 433.33General Tips: For obtaining a higher solubility , please warm…
Product Name: Refametinib R enantiomerSubtitle: MEK1/2 allosteric inhibitorBiological Activity: SMLES: COC1=CC(=C(C(=C1NS(=O)(=O)C2(CC2)CC(CO)O)NC3=C(C=C(C=C3)I)F)F)FCAS NO: 1421373-66-1Standard In CHIKey: Casein Kinase inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C19H20F3IN2O5SM.Wt: 572.34General Tips: For obtaining a higher…
Product Name: OTS964Subtitle: TOPK inhibitor,potent and selectiveBiological Activity: SMLES: C(CN(C)C)C1=CC=C(C2=C(O)C=CC3=C2C(C=CS4)=C4C(N3)=O)C=C1CAS NO: 1218778-77-8Standard In CHIKey: Aurora Kinase inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C22H22N2O2SM.Wt: 378.49General Tips: for obtaining a higher concentration:…
Product Name: OTS514Subtitle: TOPK inhibitor,highly potentBiological Activity: SMLES: NC(C)C1=CC=C(C2=C(O)C=CC3=C2C(C=CS4)=C4C(N3)=O)C=C1CAS NO: 1216941-48-8Standard In CHIKey: ATM_ATR inhibitorsStandard InChI: Typrof Compound: Appearance: Formula: C20H18N2O2SM.Wt: 350.43General Tips: For obtaining a higher solubility , please…