PD168393
Product Name: PD168393Subtitle: EGFR inhibitorBiological Activity: Biological Activity of PD168393Description PD168393 is a potent, cell-permeable, irreversible inhibitor of EGFR with IC50 value of 700 pM. Targets EGFR IC50 700 pMSMLES:…
Pelitinib (EKB-569)
Product Name: Pelitinib (EKB-569)Subtitle: EGFR inhibitor,potent and irreversibleBiological Activity: Biological Activity of Pelitinib (EKB-569)Description Pelitinib is a potent irreversible inhibitor of EGFR with IC50 value of 38.5 nM. Targets EGFR…
WZ8040
Product Name: WZ8040Subtitle: EGFR T790M inhibitor,irreversible amd potentBiological Activity: Biological Activity of WZ8040Description WZ8040 is an irreversible inhibitor of EGFR T790M with IC50 value of
WZ4002
Product Name: WZ4002Subtitle: Mutant-selective EGFR inhibitor(L858R,T790M), irreversible and potentBiological Activity: Biological Activity of WZ4002Description WZ4002 is a novel, mutant-selective inhibitor of EGFR for EGFR(L858R)/(T790M) with IC50 of 2 nM/8 nM.…
AP26113
Product Name: AP26113Subtitle: Anaplastic lymphoma kinase (ALK) inhibitorBiological Activity: Biological Activity of AP26113Description AP26113 is a potent inhibitor of ALK with IC50 of 0.62 nM. Targets ALK FER ROS/ROS1 FLT3…
AG-18
Product Name: AG-18Subtitle: EGFR/PDGFR inhibitorBiological Activity: Biological Activity of AG-18Inhibitor of epidermal growth factor receptor (EGFR) and platelet-derived growth factor receptor (PDGFR) kinase (IC50 values are 35 and 25 μM…
Gefitinib
Product Name: GefitinibSubtitle: Selective EGFR inhibitorBiological Activity: Biological Activity of Gefitinib Orally active, selective inhibitor of EGFR tyrosine kinase (IC50 = 23 – 79 nM). Shows minimal activity against ErbB2,…
Corylifol A
Product Name: Corylifol ASubtitle: Biological Activity: SMLES: CAS NO: 1155419-89-8Standard In CHIKey: Syk inhibitorsStandard InChI: Typrof Compound: FlavonoidsAppearance: Yellow powderFormula: C25H26O4M.Wt: 390.5General Tips: For obtaining a higher solubility , please…
Canertinib
Product Name: CanertinibSubtitle: HER family tyrosine kinase inhibitorBiological Activity: Biological Activity of Canertinib 1. Canertinib is a novel ErbB-receptor inhibitor currently in clinical development for the treatment of solid tumors…
Butein
Product Name: ButeinSubtitle: Protein kinase inhibitorBiological Activity: Biological Activity of Butein 1. Butein has potent anticancer activity, which includes against EGFR and MET in acquired-resistance NSCLC, ovarian cancer. 2. Butein…